RAS-inhibiting biologics identify and probe druggable pockets including an SII-α3 allosteric site
Katarzyna Z Haza, Heather L Martin, Ajinkya Rao, Amy L Turner, Sophie E Saunders, Britta Petersen, Christian Tiede, Kevin Tipping, Anna A Tang, Modupe Ajayi, Thomas Taylor, Keri M Fishwick, Thomas L Adams, Thembaninkosi G. Gaule, Chi H Trinh, Matthew Johnson, Alexander L Breeze, Thomas A Edwards, Michael J McPherson, Darren C Tomlinson
bioRxiv 2020.06.04.133728; doi: https://doi.org/10.1101/2020.06.04.133728