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Identification and Optimization of cell active 4-anilino-quin(az)oline Inhibitors for Protein Kinase Novel 3 (PKN3)
View ORCID ProfileChristopher R. M. Asquith, Louisa Temme, View ORCID ProfileTuomo Laitinen, Julie Pickett, Frank E. Kwarcinski, Parvathi Sinha, View ORCID ProfileCarrow I. Wells, View ORCID ProfileGraham J. Tizzard, Reena Zutshi, David H. Drewry
doi: https://doi.org/10.1101/2020.03.02.972943
Christopher R. M. Asquith
aDepartment of Pharmacology, School of Medicine, University of North Carolina at Chapel Hill, NC 27599, (USA)
bStructural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, NC 27599, (USA)
Louisa Temme
bStructural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, NC 27599, (USA)
Tuomo Laitinen
cSchool of Pharmacy, Faculty of Health Sciences, University of Eastern Finland, 70211 Kuopio, (Finland)
Julie Pickett
bStructural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, NC 27599, (USA)
Frank E. Kwarcinski
dLuceome Biotechnologies, LLC, Tucson, AZ 85719 (USA)
Parvathi Sinha
dLuceome Biotechnologies, LLC, Tucson, AZ 85719 (USA)
Carrow I. Wells
bStructural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, NC 27599, (USA)
Graham J. Tizzard
eSchool of Chemistry, University of Southampton, Southampton, SO17 1BJ, (United Kingdom)
Reena Zutshi
dLuceome Biotechnologies, LLC, Tucson, AZ 85719 (USA)
David H. Drewry
bStructural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, NC 27599, (USA)
Article usage
Posted March 03, 2020.
Identification and Optimization of cell active 4-anilino-quin(az)oline Inhibitors for Protein Kinase Novel 3 (PKN3)
Christopher R. M. Asquith, Louisa Temme, Tuomo Laitinen, Julie Pickett, Frank E. Kwarcinski, Parvathi Sinha, Carrow I. Wells, Graham J. Tizzard, Reena Zutshi, David H. Drewry
bioRxiv 2020.03.02.972943; doi: https://doi.org/10.1101/2020.03.02.972943
Identification and Optimization of cell active 4-anilino-quin(az)oline Inhibitors for Protein Kinase Novel 3 (PKN3)
Christopher R. M. Asquith, Louisa Temme, Tuomo Laitinen, Julie Pickett, Frank E. Kwarcinski, Parvathi Sinha, Carrow I. Wells, Graham J. Tizzard, Reena Zutshi, David H. Drewry
bioRxiv 2020.03.02.972943; doi: https://doi.org/10.1101/2020.03.02.972943
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