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Activity profiling of SARS-CoV-2-PLpro protease provides structural framework for anti-COVID-19 drug design
Wioletta Rut, Mikolaj Zmudzinski, Zongyang Lyu, Digant Nayak, Scott J. Snipas, Miklos Bekes, Tony T. Huang, Shaun K. Olsen, Marcin Drag
doi: https://doi.org/10.1101/2020.04.29.068890
Wioletta Rut
1Department of Chemical Biology and Bioimaging, Wroclaw University of Science and Technology, Wyb. Wyspianskiego 27, 50-370 Wroclaw, Poland
Mikolaj Zmudzinski
1Department of Chemical Biology and Bioimaging, Wroclaw University of Science and Technology, Wyb. Wyspianskiego 27, 50-370 Wroclaw, Poland
Zongyang Lyu
2Department of Biochemistry & Molecular Biology and Hollings Cancer Center, Medical University of South Carolina, Charleston, SC, 29425, USA
5Department of Biochemistry & Structural Biology University of Texas Health Science Center at San Antonio, San Antonio, TX, 78229 USA
Digant Nayak
2Department of Biochemistry & Molecular Biology and Hollings Cancer Center, Medical University of South Carolina, Charleston, SC, 29425, USA
5Department of Biochemistry & Structural Biology University of Texas Health Science Center at San Antonio, San Antonio, TX, 78229 USA
Scott J. Snipas
3Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, CA 92037, USA
Miklos Bekes
4Department of Biochemistry & Molecular Pharmacology, New York University School of Medicine, New York, NY 10016, USA
6Arvinas, Inc., 5 Science Park, New Haven, CT, 06511, USA
Tony T. Huang
4Department of Biochemistry & Molecular Pharmacology, New York University School of Medicine, New York, NY 10016, USA
Shaun K. Olsen
2Department of Biochemistry & Molecular Biology and Hollings Cancer Center, Medical University of South Carolina, Charleston, SC, 29425, USA
5Department of Biochemistry & Structural Biology University of Texas Health Science Center at San Antonio, San Antonio, TX, 78229 USA
Marcin Drag
1Department of Chemical Biology and Bioimaging, Wroclaw University of Science and Technology, Wyb. Wyspianskiego 27, 50-370 Wroclaw, Poland
3Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, CA 92037, USA
Article usage
Posted April 29, 2020.
Activity profiling of SARS-CoV-2-PLpro protease provides structural framework for anti-COVID-19 drug design
Wioletta Rut, Mikolaj Zmudzinski, Zongyang Lyu, Digant Nayak, Scott J. Snipas, Miklos Bekes, Tony T. Huang, Shaun K. Olsen, Marcin Drag
bioRxiv 2020.04.29.068890; doi: https://doi.org/10.1101/2020.04.29.068890
Activity profiling of SARS-CoV-2-PLpro protease provides structural framework for anti-COVID-19 drug design
Wioletta Rut, Mikolaj Zmudzinski, Zongyang Lyu, Digant Nayak, Scott J. Snipas, Miklos Bekes, Tony T. Huang, Shaun K. Olsen, Marcin Drag
bioRxiv 2020.04.29.068890; doi: https://doi.org/10.1101/2020.04.29.068890
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