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A tropane-based ibogaine analog rescues folding-deficient SERT and DAT
Shreyas Bhat, Daryl A. Guthrie, Ameya Kasture, Ali El-Kasaby, Jianjing Cao, Alessandro Bonifazi, Therese Ku, JoLynn B. Giancola, Thomas Hummel, View ORCID ProfileMichael Freissmuth, Amy Hauck Newman
doi: https://doi.org/10.1101/2020.07.14.202325
Shreyas Bhat
1Institute of Pharmacology and the Gaston H. Glock Research Laboratories for Exploratory Drug Development, Center of Physiology and Pharmacology, Medical University of Vienna, Vienna, Waehringerstrasse 13a, Vienna, Austria
Daryl A. Guthrie
2Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse, Intramural Research Program, Baltimore, MD 21224, U.S.A
Ameya Kasture
3Department of Neurobiology, University of Vienna, Austria
Ali El-Kasaby
1Institute of Pharmacology and the Gaston H. Glock Research Laboratories for Exploratory Drug Development, Center of Physiology and Pharmacology, Medical University of Vienna, Vienna, Waehringerstrasse 13a, Vienna, Austria
Jianjing Cao
2Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse, Intramural Research Program, Baltimore, MD 21224, U.S.A
Alessandro Bonifazi
2Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse, Intramural Research Program, Baltimore, MD 21224, U.S.A
Therese Ku
2Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse, Intramural Research Program, Baltimore, MD 21224, U.S.A
JoLynn B. Giancola
2Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse, Intramural Research Program, Baltimore, MD 21224, U.S.A
Thomas Hummel
3Department of Neurobiology, University of Vienna, Austria
Michael Freissmuth
1Institute of Pharmacology and the Gaston H. Glock Research Laboratories for Exploratory Drug Development, Center of Physiology and Pharmacology, Medical University of Vienna, Vienna, Waehringerstrasse 13a, Vienna, Austria
Amy Hauck Newman
2Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse, Intramural Research Program, Baltimore, MD 21224, U.S.A
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Posted July 14, 2020.
A tropane-based ibogaine analog rescues folding-deficient SERT and DAT
Shreyas Bhat, Daryl A. Guthrie, Ameya Kasture, Ali El-Kasaby, Jianjing Cao, Alessandro Bonifazi, Therese Ku, JoLynn B. Giancola, Thomas Hummel, Michael Freissmuth, Amy Hauck Newman
bioRxiv 2020.07.14.202325; doi: https://doi.org/10.1101/2020.07.14.202325
A tropane-based ibogaine analog rescues folding-deficient SERT and DAT
Shreyas Bhat, Daryl A. Guthrie, Ameya Kasture, Ali El-Kasaby, Jianjing Cao, Alessandro Bonifazi, Therese Ku, JoLynn B. Giancola, Thomas Hummel, Michael Freissmuth, Amy Hauck Newman
bioRxiv 2020.07.14.202325; doi: https://doi.org/10.1101/2020.07.14.202325
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