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Identification, Characterization and Synthesis of Natural Parasitic Cysteine Protease Inhibitors – More Potent Falcitidin Analogs
View ORCID ProfileStephan Brinkmann, Sandra Semmler, View ORCID ProfileChristian Kersten, View ORCID ProfileMaria A. Patras, Michael Kurz, View ORCID ProfileNatalie Fuchs, View ORCID ProfileStefan J. Hammerschmidt, Jennifer Legac, Peter E. Hammann, View ORCID ProfileAndreas Vilcinskas, View ORCID ProfilePhilip. J. Rosenthal, View ORCID ProfileTanja Schirmeister, View ORCID ProfileArmin Bauer, View ORCID ProfileTill F. Schäberle
doi: https://doi.org/10.1101/2021.10.30.466580
Stephan Brinkmann
1Fraunhofer Institute for Molecular Biology and Applied Ecology (IME), Branch for Bioresources, 35392 Giessen, Germany
Sandra Semmler
1Fraunhofer Institute for Molecular Biology and Applied Ecology (IME), Branch for Bioresources, 35392 Giessen, Germany
Christian Kersten
2Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, 55128 Mainz, Germany
Maria A. Patras
1Fraunhofer Institute for Molecular Biology and Applied Ecology (IME), Branch for Bioresources, 35392 Giessen, Germany
Michael Kurz
3Sanofi-Aventis Deutschland GmbH, R&D, 65926 Frankfurt am Main, Germany
Natalie Fuchs
2Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, 55128 Mainz, Germany
Stefan J. Hammerschmidt
2Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, 55128 Mainz, Germany
Jennifer Legac
4Department of Medicine, University of California, San Francisco, 94143 California, United States
Peter E. Hammann
5Evotec International GmbH, 37079 Göttingen, Germany
Andreas Vilcinskas
1Fraunhofer Institute for Molecular Biology and Applied Ecology (IME), Branch for Bioresources, 35392 Giessen, Germany
6Institute for Insect Biotechnology, Justus-Liebig-University of Giessen, 35392 Giessen, Germany
Philip. J. Rosenthal
4Department of Medicine, University of California, San Francisco, 94143 California, United States
Tanja Schirmeister
2Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, 55128 Mainz, Germany
Armin Bauer
3Sanofi-Aventis Deutschland GmbH, R&D, 65926 Frankfurt am Main, Germany
Till F. Schäberle
1Fraunhofer Institute for Molecular Biology and Applied Ecology (IME), Branch for Bioresources, 35392 Giessen, Germany
6Institute for Insect Biotechnology, Justus-Liebig-University of Giessen, 35392 Giessen, Germany
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Posted October 30, 2021.
Identification, Characterization and Synthesis of Natural Parasitic Cysteine Protease Inhibitors – More Potent Falcitidin Analogs
Stephan Brinkmann, Sandra Semmler, Christian Kersten, Maria A. Patras, Michael Kurz, Natalie Fuchs, Stefan J. Hammerschmidt, Jennifer Legac, Peter E. Hammann, Andreas Vilcinskas, Philip. J. Rosenthal, Tanja Schirmeister, Armin Bauer, Till F. Schäberle
bioRxiv 2021.10.30.466580; doi: https://doi.org/10.1101/2021.10.30.466580
Identification, Characterization and Synthesis of Natural Parasitic Cysteine Protease Inhibitors – More Potent Falcitidin Analogs
Stephan Brinkmann, Sandra Semmler, Christian Kersten, Maria A. Patras, Michael Kurz, Natalie Fuchs, Stefan J. Hammerschmidt, Jennifer Legac, Peter E. Hammann, Andreas Vilcinskas, Philip. J. Rosenthal, Tanja Schirmeister, Armin Bauer, Till F. Schäberle
bioRxiv 2021.10.30.466580; doi: https://doi.org/10.1101/2021.10.30.466580
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