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Targeting a Therapy-Resistant Cancer Cell State Using Masked Electrophiles as GPX4 Inhibitors
View ORCID ProfileJohn K. Eaton, Laura Furst, Richard A. Ruberto, Dieter Moosmayer, Roman C. Hillig, André Hilpmann, Katja Zimmermann, Matthew J. Ryan, Michael Niehues, Volker Badock, Anneke Kramm, Sixun Chen, Paul A. Clemons, Stefan Gradl, Claire Montagnon, Kiel E. Lazarski, Sven Christian, Besnik Bajrami, Roland Neuhaus, Ashley L. Eheim, View ORCID ProfileVasanthi S. Viswanathan, View ORCID ProfileStuart L. Schreiber
doi: https://doi.org/10.1101/376764
John K. Eaton
1Broad Institute, Cambridge, MA 02142, USA
Laura Furst
1Broad Institute, Cambridge, MA 02142, USA
Richard A. Ruberto
1Broad Institute, Cambridge, MA 02142, USA
Dieter Moosmayer
2Bayer AG, Berlin 13353, Germany
Roman C. Hillig
2Bayer AG, Berlin 13353, Germany
André Hilpmann
2Bayer AG, Berlin 13353, Germany
Katja Zimmermann
2Bayer AG, Berlin 13353, Germany
Matthew J. Ryan
1Broad Institute, Cambridge, MA 02142, USA
Michael Niehues
2Bayer AG, Berlin 13353, Germany
Volker Badock
2Bayer AG, Berlin 13353, Germany
Anneke Kramm
1Broad Institute, Cambridge, MA 02142, USA
Sixun Chen
1Broad Institute, Cambridge, MA 02142, USA
Paul A. Clemons
1Broad Institute, Cambridge, MA 02142, USA
Stefan Gradl
2Bayer AG, Berlin 13353, Germany
Claire Montagnon
1Broad Institute, Cambridge, MA 02142, USA
Kiel E. Lazarski
1Broad Institute, Cambridge, MA 02142, USA
Sven Christian
2Bayer AG, Berlin 13353, Germany
Besnik Bajrami
1Broad Institute, Cambridge, MA 02142, USA
Roland Neuhaus
2Bayer AG, Berlin 13353, Germany
Ashley L. Eheim
2Bayer AG, Berlin 13353, Germany
Vasanthi S. Viswanathan
1Broad Institute, Cambridge, MA 02142, USA
Stuart L. Schreiber
1Broad Institute, Cambridge, MA 02142, USA
3Department of Chemistry and Chemical Biology, Harvard University, Cambridge, MA 02138, USA
4Howard Hughes Medical Institute, Cambridge, MA 02138, USA
Article usage
Posted September 05, 2018.
Targeting a Therapy-Resistant Cancer Cell State Using Masked Electrophiles as GPX4 Inhibitors
John K. Eaton, Laura Furst, Richard A. Ruberto, Dieter Moosmayer, Roman C. Hillig, André Hilpmann, Katja Zimmermann, Matthew J. Ryan, Michael Niehues, Volker Badock, Anneke Kramm, Sixun Chen, Paul A. Clemons, Stefan Gradl, Claire Montagnon, Kiel E. Lazarski, Sven Christian, Besnik Bajrami, Roland Neuhaus, Ashley L. Eheim, Vasanthi S. Viswanathan, Stuart L. Schreiber
bioRxiv 376764; doi: https://doi.org/10.1101/376764
Targeting a Therapy-Resistant Cancer Cell State Using Masked Electrophiles as GPX4 Inhibitors
John K. Eaton, Laura Furst, Richard A. Ruberto, Dieter Moosmayer, Roman C. Hillig, André Hilpmann, Katja Zimmermann, Matthew J. Ryan, Michael Niehues, Volker Badock, Anneke Kramm, Sixun Chen, Paul A. Clemons, Stefan Gradl, Claire Montagnon, Kiel E. Lazarski, Sven Christian, Besnik Bajrami, Roland Neuhaus, Ashley L. Eheim, Vasanthi S. Viswanathan, Stuart L. Schreiber
bioRxiv 376764; doi: https://doi.org/10.1101/376764
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