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A Chemical Toolbox for the Study of Bromodomains and Epigenetic Signaling
Qin Wu, David Heidenreich, Stanley Zhou, Suzanne Ackloo, Genevieve Deblois, Shili Duan, Kiran Nakka, Jeffrey Dilworth, Mathieu Lupien, Paul E. Brennan, Cheryl H. Arrowsmith, Susanne Müller, Oleg Fedorov, Panagis Filippakopoulos, Stefan Knapp
doi: https://doi.org/10.1101/391870
Qin Wu
2Structural Genomics Consortium, University of Toronto, Toronto, Ontario, M5G 1L7, Canada
3Princess Margaret Cancer Centre, University Health Network, Toronto, Ontario, Canada
4Department of Medical Biophysics, University of Toronto, Toronto M5G 2M9, ON, Canada
David Heidenreich
11nstitute of Pharmaceutical Chemistry, Goethe-University Frankfurt, 60438 Frankfurt, Germany
6Structural Genomics Consortium, Buchmann Institute for Life Sciences, Goethe-University Frankfurt, 60438 Frankfurt, Germany
Stanley Zhou
3Princess Margaret Cancer Centre, University Health Network, Toronto, Ontario, Canada
4Department of Medical Biophysics, University of Toronto, Toronto M5G 2M9, ON, Canada
Suzanne Ackloo
2Structural Genomics Consortium, University of Toronto, Toronto, Ontario, M5G 1L7, Canada
Genevieve Deblois
3Princess Margaret Cancer Centre, University Health Network, Toronto, Ontario, Canada
4Department of Medical Biophysics, University of Toronto, Toronto M5G 2M9, ON, Canada
Shili Duan
3Princess Margaret Cancer Centre, University Health Network, Toronto, Ontario, Canada
4Department of Medical Biophysics, University of Toronto, Toronto M5G 2M9, ON, Canada
Kiran Nakka
9Sprott Centre for Stem Cell Research, Regenerative Medicine Program, Ottawa Hospital Research Institute, Ottawa, Canada
Jeffrey Dilworth
9Sprott Centre for Stem Cell Research, Regenerative Medicine Program, Ottawa Hospital Research Institute, Ottawa, Canada
Mathieu Lupien
3Princess Margaret Cancer Centre, University Health Network, Toronto, Ontario, Canada
4Department of Medical Biophysics, University of Toronto, Toronto M5G 2M9, ON, Canada
Paul E. Brennan
8Target Discovery Institute and Structural Genomics Consortium, University of Oxford, Oxford OX3 7DQ, UK
Cheryl H. Arrowsmith
2Structural Genomics Consortium, University of Toronto, Toronto, Ontario, M5G 1L7, Canada
3Princess Margaret Cancer Centre, University Health Network, Toronto, Ontario, Canada
4Department of Medical Biophysics, University of Toronto, Toronto M5G 2M9, ON, Canada
Susanne Müller
11nstitute of Pharmaceutical Chemistry, Goethe-University Frankfurt, 60438 Frankfurt, Germany
6Structural Genomics Consortium, Buchmann Institute for Life Sciences, Goethe-University Frankfurt, 60438 Frankfurt, Germany
Oleg Fedorov
8Target Discovery Institute and Structural Genomics Consortium, University of Oxford, Oxford OX3 7DQ, UK
Panagis Filippakopoulos
8Target Discovery Institute and Structural Genomics Consortium, University of Oxford, Oxford OX3 7DQ, UK
Stefan Knapp
11nstitute of Pharmaceutical Chemistry, Goethe-University Frankfurt, 60438 Frankfurt, Germany
6Structural Genomics Consortium, Buchmann Institute for Life Sciences, Goethe-University Frankfurt, 60438 Frankfurt, Germany
7German Cancer Network (DKTK), Frankfurt/Mainz, 60438 Frankfurt, Germany
Posted August 14, 2018.
A Chemical Toolbox for the Study of Bromodomains and Epigenetic Signaling
Qin Wu, David Heidenreich, Stanley Zhou, Suzanne Ackloo, Genevieve Deblois, Shili Duan, Kiran Nakka, Jeffrey Dilworth, Mathieu Lupien, Paul E. Brennan, Cheryl H. Arrowsmith, Susanne Müller, Oleg Fedorov, Panagis Filippakopoulos, Stefan Knapp
bioRxiv 391870; doi: https://doi.org/10.1101/391870
A Chemical Toolbox for the Study of Bromodomains and Epigenetic Signaling
Qin Wu, David Heidenreich, Stanley Zhou, Suzanne Ackloo, Genevieve Deblois, Shili Duan, Kiran Nakka, Jeffrey Dilworth, Mathieu Lupien, Paul E. Brennan, Cheryl H. Arrowsmith, Susanne Müller, Oleg Fedorov, Panagis Filippakopoulos, Stefan Knapp
bioRxiv 391870; doi: https://doi.org/10.1101/391870
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