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Activation loop dynamics are controlled by conformation-selective inhibitors of ERK2
View ORCID ProfileLaurel M. Pegram, Jennifer C. Liddle, Yao Xiao, Maria Hoh, View ORCID ProfileJohannes Rudolph, Dylan B. Iverson, View ORCID ProfileGuy P. Vigers, Darin Smith, Hailong Zhang, Weiru Wang, John G. Moffat, View ORCID ProfileNatalie G. Ahn
doi: https://doi.org/10.1101/639567
Laurel M. Pegram
*Department of Biochemistry, University of Colorado, Boulder, CO 80305
Jennifer C. Liddle
*Department of Biochemistry, University of Colorado, Boulder, CO 80305
Yao Xiao
*Department of Biochemistry, University of Colorado, Boulder, CO 80305
Maria Hoh
*Department of Biochemistry, University of Colorado, Boulder, CO 80305
Johannes Rudolph
*Department of Biochemistry, University of Colorado, Boulder, CO 80305
Dylan B. Iverson
*Department of Biochemistry, University of Colorado, Boulder, CO 80305
Guy P. Vigers
†Array BioPharma Inc., 3200 Walnut St., Boulder, CO, 80301
Darin Smith
†Array BioPharma Inc., 3200 Walnut St., Boulder, CO, 80301
Hailong Zhang
†Array BioPharma Inc., 3200 Walnut St., Boulder, CO, 80301
Weiru Wang
‡Genentech, Inc., 1 DNA Way, South San Francisco, CA, 94080.
John G. Moffat
‡Genentech, Inc., 1 DNA Way, South San Francisco, CA, 94080.
Natalie G. Ahn
*Department of Biochemistry, University of Colorado, Boulder, CO 80305
Article usage
Posted May 16, 2019.
Activation loop dynamics are controlled by conformation-selective inhibitors of ERK2
Laurel M. Pegram, Jennifer C. Liddle, Yao Xiao, Maria Hoh, Johannes Rudolph, Dylan B. Iverson, Guy P. Vigers, Darin Smith, Hailong Zhang, Weiru Wang, John G. Moffat, Natalie G. Ahn
bioRxiv 639567; doi: https://doi.org/10.1101/639567
Activation loop dynamics are controlled by conformation-selective inhibitors of ERK2
Laurel M. Pegram, Jennifer C. Liddle, Yao Xiao, Maria Hoh, Johannes Rudolph, Dylan B. Iverson, Guy P. Vigers, Darin Smith, Hailong Zhang, Weiru Wang, John G. Moffat, Natalie G. Ahn
bioRxiv 639567; doi: https://doi.org/10.1101/639567
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