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Table representation of search results timeline featuring number of search results per year.

Year Number of Results
1990 1
2000 1
2002 1
2003 2
2004 4
2005 7
2006 5
2007 3
2008 2
2009 2
2010 1
2011 5
2012 2
2013 2
2015 2
2017 1
2018 1
2020 4
2021 1
2023 2
2024 1

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Page 1
Systematic Chemogenetic Library Assembly.
Canham SM, Wang Y, Cornett A, Auld DS, Baeschlin DK, Patoor M, Skaanderup PR, Honda A, Llamas L, Wendel G, Mapa FA, Aspesi P Jr, Labbé-Giguère N, Gamber GG, Palacios DS, Schuffenhauer A, Deng Z, Nigsch F, Frederiksen M, Bushell SM, Rothman D, Jain RK, Hemmerle H, Briner K, Porter JA, Tallarico JA, Jenkins JL. Canham SM, et al. Among authors: schuffenhauer a. Cell Chem Biol. 2020 Sep 17;27(9):1124-1129. doi: 10.1016/j.chembiol.2020.07.004. Epub 2020 Jul 23. Cell Chem Biol. 2020. PMID: 32707038 Free article. Review.
Evolution of Novartis' Small Molecule Screening Deck Design.
Schuffenhauer A, Schneider N, Hintermann S, Auld D, Blank J, Cotesta S, Engeloch C, Fechner N, Gaul C, Giovannoni J, Jansen J, Joslin J, Krastel P, Lounkine E, Manchester J, Monovich LG, Pelliccioli AP, Schwarze M, Shultz MD, Stiefl N, Baeschlin DK. Schuffenhauer A, et al. J Med Chem. 2020 Dec 10;63(23):14425-14447. doi: 10.1021/acs.jmedchem.0c01332. Epub 2020 Nov 3. J Med Chem. 2020. PMID: 33140646 Review.
Library design for fragment based screening.
Schuffenhauer A, Ruedisser S, Marzinzik AL, Jahnke W, Blommers M, Selzer P, Jacoby E. Schuffenhauer A, et al. Curr Top Med Chem. 2005;5(8):751-62. doi: 10.2174/1568026054637700. Curr Top Med Chem. 2005. PMID: 16101415 Review.
Complex molecules: do they add value?
Selzer P, Roth HJ, Ertl P, Schuffenhauer A. Selzer P, et al. Among authors: schuffenhauer a. Curr Opin Chem Biol. 2005 Jun;9(3):310-6. doi: 10.1016/j.cbpa.2005.04.001. Curr Opin Chem Biol. 2005. PMID: 15939334 Review.
N-aryl-piperidine-4-carboxamides as a novel class of potent inhibitors of MALT1 proteolytic activity.
Schlapbach A, Revesz L, Pissot Soldermann C, Zoller T, Régnier CH, Bornancin F, Radimerski T, Blank J, Schuffenhauer A, Renatus M, Erbel P, Melkko S, Heng R, Simic O, Endres R, Wartmann M, Quancard J. Schlapbach A, et al. Among authors: schuffenhauer a. Bioorg Med Chem Lett. 2018 Jul 1;28(12):2153-2158. doi: 10.1016/j.bmcl.2018.05.017. Epub 2018 May 9. Bioorg Med Chem Lett. 2018. PMID: 29759726
Latent hit series hidden in high-throughput screening data.
Varin T, Didiot MC, Parker CN, Schuffenhauer A. Varin T, et al. Among authors: schuffenhauer a. J Med Chem. 2012 Feb 9;55(3):1161-70. doi: 10.1021/jm201328e. Epub 2012 Jan 23. J Med Chem. 2012. PMID: 22185196
46 results