A data set consisting of twenty-two sertindole analogues and ten structurally diverse inhibitors,
spanning a wide range in potency, was analyzed using CoMSiA. A homology model of …

A comprehensive comparative analysis of the structure-antifungal activity relationships for
the series of biosynthetically engineered nystatin analogues and their novel semisynthetic …

Solid-state NMR has been used to examine isolated cell walls and intact whole cells of
Staphylococcus aureus complexed to five different vancomycin, eremomycin, and …

Anthraquinones and their analogues, in particular heteroarene-fused anthracendiones, are
prospective scaffolds for new compounds with improved antitumor characteristics. We herein …

… Maria N. Preobrazhenskaya, a brilliant scientist and wonderful colleague who initiated our
productive … We would like to thank members of both the Firestone and the Preobrazhenskaya …

A variety of semisynthetic derivatives of natural antibacterial glycopeptide antibiotics such
as vancomycin, eremomycin, ristocetin A, teicoplanin A 2 -2, DA-40926, their aglycons, and …

Various semisynthetic derivatives of glycopeptide antibiotics including vancomycin, eremomycin,
teicoplanin, ristocetin A and DA-40926 have been evaluated for their inhibitory activity …

Antiviral activity and other biological properties of two groups of polycyclic peptides are
discussed. Antibiotics of the complestatin–kistamycin group have a structural motif similar to that …

We developed the synthesis of a series of thiophene-fused tetracyclic analogues of the
antitumor drug ametantrone. The reactions included nucleophilic substitution of methoxy groups …

There is an urgent need for potent inhibitors of dengue virus (DENV) replication for the treatment
and/or prophylaxis of infections with this virus. We here report on an aglycon analogue …